6HTR |
Yeast 20S proteasome with human beta2c (S171G) in complex with 13 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/04/2018 |
2.6 |
0.1937 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae S288c |
X-RAY DIFFRACTION |
1 |
6HTB |
Yeast 20S proteasome with human beta2c (S171G) |
HYDROLASE |
HYDROLASE, Proteasome, Mutant |
10/03/2018 |
2.7 |
0.19265 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae S288c |
X-RAY DIFFRACTION |
1 |
6HVA |
Yeast 20S proteasome with human beta2i (1-53) in complex with 13 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/10/2018 |
2.9 |
0.18184 |
Saccharomyces cerevisiae S288C |
Saccharomyces cerevisiae S288C |
X-RAY DIFFRACTION |
1 |
6HV5 |
Yeast 20S proteasome with human beta2i (1-53) in complex with 4 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/10/2018 |
3.0 |
0.17331 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae S288C |
X-RAY DIFFRACTION |
1 |
6HV4 |
Yeast 20S proteasome with human beta2i (1-53) in complex with ONX 0914 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/10/2018 |
3.0 |
0.18379 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HUV |
Yeast 20S proteasome with human beta2c (S171G) in complex with 39 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/09/2018 |
3.1 |
0.1683 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HV7 |
Yeast 20S proteasome with human beta2i (1-53) in complex with 7 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/10/2018 |
3.4 |
0.1737 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae S288c |
X-RAY DIFFRACTION |
1 |
6HUU |
Yeast 20S proteasome with human beta2c (S171G) in complex with 29 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/09/2018 |
2.8 |
0.19438 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HV3 |
Yeast 20S proteasome with human beta2i (1-53) |
HYDROLASE |
HYDROLASE, Proteasome, Mutant |
10/10/2018 |
2.7 |
0.17669 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HUQ |
Yeast 20S proteasome with human beta2c (S171G) in complex with 20 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/09/2018 |
3.0 |
0.17796 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HUC |
Yeast 20S proteasome with human beta2c (S171G) in complex with 18 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/05/2018 |
3.0 |
0.18144 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae |
X-RAY DIFFRACTION |
1 |
6HWD |
Yeast 20S proteasome beta2-G45A mutant in complex with bortezomib |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/11/2018 |
2.8 |
0.18589 |
Saccharomyces cerevisiae S288c |
Saccharomyces cerevisiae S288c |
X-RAY DIFFRACTION |
1 |
6HWC |
Yeast 20S proteasome beta2-G45A mutant |
HYDROLASE |
Proteasome, Mutant, HYDROLASE |
10/11/2018 |
2.8 |
0.195 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
— |
X-RAY DIFFRACTION |
1 |
6HVU |
Yeast 20S proteasome with human beta2i (1-53) in complex with 29 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/11/2018 |
2.9 |
0.18964 |
Saccharomyces cerevisiae S288C |
Saccharomyces cerevisiae S288C |
X-RAY DIFFRACTION |
1 |
6HW6 |
Yeast 20S proteasome in complex with 20 |
HYDROLASE |
HYDROLASE, Proteasome, Inhibitor, Binding Analysis |
10/11/2018 |
2.7 |
0.17517 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
— |
X-RAY DIFFRACTION |
1 |
6HVT |
Yeast 20S proteasome with human beta2i (1-53) in complex with 20 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/11/2018 |
2.9 |
0.1792 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
X-RAY DIFFRACTION |
1 |
6HVW |
Yeast 20S proteasome with human beta2i (1-53) in complex with 43 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/11/2018 |
3.0 |
0.16461 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
Saccharomyces cerevisiae S288c |
X-RAY DIFFRACTION |
1 |
6HVV |
Yeast 20S proteasome with human beta2i (1-53) in complex with 39 |
HYDROLASE |
Proteasome, Mutant, Inhibitor, Binding Analysis, HYDROLASE |
10/11/2018 |
2.7 |
0.18419 |
Saccharomyces cerevisiae S288C |
Saccharomyces cerevisiae S288C |
X-RAY DIFFRACTION |
1 |
6HVY |
Yeast 20S proteasome in complex with 5 (7- and 6-membered ring) |
HYDROLASE |
HYDROLASE, Proteasome, Inhibitor, Binding Analysis |
10/11/2018 |
2.7 |
0.18145 |
Saccharomyces cerevisiae (strain ATCC 204508 / S288c) |
— |
X-RAY DIFFRACTION |
1 |
7AKS |
Human ADP-ribosylserine hydrolase ARH3 mutant E41A in complex with H2B-S7-mar peptide |
HYDROLASE |
ADP-RIBOSYLATION, ADP-RIBOSE, ADPRHL2, ADP-RIBOSYLHYDROLASE LIKE 2, SER-ADPR, SERINE-ADPR, ADP-RIBOSYL-L-SERINE, HYDROLASE |
10/02/2020 |
1.86 |
0.1685 |
Homo sapiens |
Escherichia coli |
X-RAY DIFFRACTION |
2 |